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Cariprazine HCl
CAS No. 1083076-69-0
Cariprazine HCl ( RGH188 hydrochloride )
产品货号. M21610 CAS No. 1083076-69-0
Cariprazine HCl is an antipsychotic drug is a D3 and D2?receptor partial agonist((Ki of 0.085 nM and 0.49 nM respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | ￥616 | 有现货 |
|
| 50MG | ￥940 | 有现货 |
|
| 100MG | ￥1401 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Cariprazine HCl
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Cariprazine HCl is an antipsychotic drug is a D3 and D2?receptor partial agonist((Ki of 0.085 nM and 0.49 nM respectively).
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产品描述Cariprazine HCl is an antipsychotic drug is a D3 and D2?receptor partial agonist((Ki of 0.085 nM and 0.49 nM respectively).
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同义词RGH188 hydrochloride
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通路GPCR/G Protein
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靶点Dopamine Receptor
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受体D2;D3
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研究领域Neurological Disease
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适应症Major Depressive Disorder
化学信息
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CAS Number1083076-69-0
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分子量463.87
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分子式C21H33Cl3N4O
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纯度>98% (HPLC)
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溶解度DMSO:6.67 mg/mL (14.38 mM; Need ultrasonic)
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SMILESCl.CN(C)C(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)c2cccc(Cl)c2Cl)CC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Seneca N et al. Occupancy of dopamine D2 and D3 and serotonin 5-HT1A receptors by the novel antipsychotic drug candidate cariprazine (RGH-188) in monkey brain measured using positron emission tomography. Psychopharmacology (Berl). 2011 Dec;218(3):579-8
产品手册
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